Properidine
Chemical compound
- none
- AU: S9 (Prohibited substance)
- BR: Class A1 (Narcotic drugs)[1]
- CA: Schedule I
- DE: Anlage I (Authorized scientific use only)
- UK: Class A
- US: Schedule I
- UN: Psychotropic Schedule I
- isopropyl 1-methyl-4-phenylpiperidine-4-carboxylate
- 561-76-2 N
- 62373
- 56161 Y
- R1493W1CJ0
- DTXSID20204644
- Interactive image
- O=C(OC(C)C)C2(c1ccccc1)CCN(C)CC2
InChI
- InChI=1S/C16H23NO2/c1-13(2)19-15(18)16(9-11-17(3)12-10-16)14-7-5-4-6-8-14/h4-8,13H,9-12H2,1-3H3 Y
- Key:XJKQCILVUHXVIQ-UHFFFAOYSA-N Y
Properidine is an opioid, an analgesic, and the isopropyl analog of pethidine.[2] Properidine is under international control and is listed in the United States under the Controlled Substances Act (1970) as a Schedule I substance. It is a narcotic, with an Administrative Controlled Substances Code Number (ACSCN) of 9644 and a 2 gramme annual aggregate manufacturing quota as of 2014. The salt in use is hydrochloride, with a free base conversion ratio of 0.88.[3]
References
- ^ Anvisa (2023-03-31). "RDC Nº 784 - Listas de Substâncias Entorpecentes, Psicotrópicas, Precursoras e Outras sob Controle Especial" [Collegiate Board Resolution No. 784 - Lists of Narcotic, Psychotropic, Precursor, and Other Substances under Special Control] (in Brazilian Portuguese). Diário Oficial da União (published 2023-04-04). Archived from the original on 2023-08-03. Retrieved 2023-08-16.
- ^ Morrison AL, Rinderknecht H (1950). "302. Synthetic analgesics. Part V. Compounds related to pethidine". Journal of the Chemical Society (Resumed): 1467. doi:10.1039/JR9500001467.
- ^ "Quotas - 2014". Diversion Control Division. U.S. Department of Justice, Drug Enforcement Administration.
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Antagonists |
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- Enkephalinase inhibitors: Amastatin
- BL-2401
- Candoxatril
- D -Phenylalanine
- Dexecadotril (retorphan)
- Ecadotril (sinorphan)
- Kelatorphan
- Racecadotril (acetorphan)
- RB-101
- RB-120
- RB-3007
- Opiorphan
- Selank
- Semax
- Spinorphin
- Thiorphan
- Tynorphin
- Ubenimex (bestatin)
- Propeptides: β-Lipotropin (proendorphin)
- Prodynorphin
- Proenkephalin
- Pronociceptin
- Proopiomelanocortin (POMC)
- Others: Kyotorphin (met-enkephalin releaser/degradation stabilizer)
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