14-Ethoxymetopon
Chemical compound
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Formula | C20H25NO4 |
Molar mass | 343.423 g·mol−1 |
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14-Ethoxymetopon[1] is an opioid analog that is a derivative of metopon which has been substituted with an ethoxy group at the 14-position. It is a highly potent analgesic drug several hundred times more potent than morphine.[2]
References
- ^ US 6476044, Wnendt S, Strassburger W, Buschmann H, Reiss-Mueller E, Krueger T, "Use of morphine derivatives as medicaments for the treatment of neuropathic problems", published 2002-11-07
- ^ Fürst Z, Búzás B, Friedmann T, Schmidhammer H, Borsodi A (May 1993). "Highly potent novel opioid receptor agonist in the 14-alkoxymetopon series". European Journal of Pharmacology. 236 (2): 209–15. doi:10.1016/0014-2999(93)90591-5. PMID 8391457.
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Opioid receptor modulators
(MOR)
(DOR)
(KOR)
(NOP)
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Antagonists |
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- Enkephalinase inhibitors: Amastatin
- BL-2401
- Candoxatril
- D -Phenylalanine
- Dexecadotril (retorphan)
- Ecadotril (sinorphan)
- Kelatorphan
- Racecadotril (acetorphan)
- RB-101
- RB-120
- RB-3007
- Opiorphan
- Selank
- Semax
- Spinorphin
- Thiorphan
- Tynorphin
- Ubenimex (bestatin)
- Propeptides: β-Lipotropin (proendorphin)
- Prodynorphin
- Proenkephalin
- Pronociceptin
- Proopiomelanocortin (POMC)
- Others: Kyotorphin (met-enkephalin releaser/degradation stabilizer)
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